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1,3-DIPOLAR CYCLOADDITION OF PYRIDYNES AND AZIDES: CONCISE SYNTHESIS OF TRIAZOLOPYRIDINES
| Title: | 1,3-DIPOLAR CYCLOADDITION OF PYRIDYNES AND AZIDES: CONCISE SYNTHESIS OF TRIAZOLOPYRIDINES |
| Authors: | Saito, Nozomi Browse this author →KAKEN DB | | Nakamura, Ken-ichi Browse this author | | Sato, Yoshihiro Browse this author →KAKEN DB |
| Issue Date: | 1-Jan-2014 |
| Publisher: | Pergamon-elsevier science ltd |
| Journal Title: | Heterocycles |
| Volume: | 88 |
| Issue: | 2 |
| Start Page: | 929 |
| End Page: | 937 |
| Publisher DOI: | 10.3987/COM-13-S(S)86 |
| Abstract: | 1,3-Dipolar cycloaddition of pyridynes and organic azides was investigated. Thus, 3,4-pyridynes and 2,3-pyridynes were reacted with various organic azides under mild conditions to afford the corresponding [1,2,3]triazolo[4,5-c]pyridines and [1,2,3]triazolo[4,5-b]pyridines, respectively. In the case of the reaction of 3,4-pyridyne, it was also found that a substituent on the pyridine ring affected the regioselectivity of the cycloaddition. |
| Type: | article (author version) |
| URI: | http://hdl.handle.net/2115/54873 |
| Appears in Collections: | 薬学研究院 (Faculty of Pharmaceutical Sciences) > 雑誌発表論文等 (Peer-reviewed Journal Articles, etc)
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Submitter: 佐藤 美洋
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